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Crystal structure of PDK1 in complex with a pyrazoloquinazoline inhibitor

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Protein Data Bank Japan2024-11-13 更新2026-03-21 收录
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Crystal structure of PDK1 in complex with a pyrazoloquinazoline inhibitor Descriptor: 3-PHOSPHOINOSITIDE DEPENDENT PROTEIN KINASE 1, 8-(CYCLOHEXA-2,5-DIEN-1-YLIDENEAMINO)-1-(PIPERIDIN-4-YLMETHYL)-4,5-DIHYDRO-1H-PYRAZOLO[4,3-H]QUINAZOLINE-3-CARBOXAMIDE, GLYCEROL, ... Authors: Angiolini, M, Banfi, P, Casale, E, Casuscelli, F, Fiorelli, C, Saccardo, M.B, Silvagni, M, Zuccotto, F. Deposit date: 2010-04-23 Release date: 2010-07-28 Last modified: 2024-11-13 Method: X-RAY DIFFRACTION (2 Å) Cite: Structure-Based Optimization of Potent Pdk1 Inhibitors. Bioorg.Med.Chem.Lett., 20, 2010
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2010-04-23
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