RIP2K kinase domain dimer with bound compound 37 (N399), a speific NOD1 pathway inhibitor
收藏Protein Data Bank Japan2024-11-27 更新2026-04-25 收录
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RIP2K kinase domain dimer with bound compound 37 (N399), a speific NOD1 pathway inhibitor Descriptor: N-[2,4-bis(chloranyl)-5-methoxy-phenyl]-7-[2-(diethylamino)ethoxy]-6-methoxy-quinazolin-4-amine, Receptor-interacting serine/threonine-protein kinase 2 Authors: Cusack, S, Huard, K, Pellegrini, E. Deposit date: 2024-04-26 Release date: 2024-11-06 Last modified: 2024-11-27 Method: X-RAY DIFFRACTION (1.943 Å) Cite: 4-Anilinoquinazoline Derivatives as the First Potent NOD1-RIPK2 Signaling Pathway Inhibitors at the Nanomolar Range. J.Med.Chem., 67, 2024
创建时间:
2024-04-26



