Crystal structure of BACE1 in complex with aminoquinoline compound 1
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Crystal structure of BACE1 in complex with aminoquinoline compound 1 Descriptor: (2R)-3-[2-amino-6-(3-methylpyridin-2-yl)quinolin-3-yl]-N-(3,3-dimethylbutyl)-2-methylpropanamide, Beta-secretase 1, GLYCEROL, ... Authors: Whittington, D.A, Long, A.M. Deposit date: 2016-02-11 Release date: 2016-03-30 Last modified: 2024-11-06 Method: X-RAY DIFFRACTION (1.62 Å) Cite: Fragment-Linking Approach Using (19)F NMR Spectroscopy To Obtain Highly Potent and Selective Inhibitors of beta-Secretase. J.Med.Chem., 59, 2016
创建时间:
2016-02-11



