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CDK2 with EGFR inhibitor compound 8

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Protein Data Bank Japan2024-11-06 更新2026-03-21 收录
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https://pdbj.org/mine/summary/4rj3
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CDK2 with EGFR inhibitor compound 8 Descriptor: 1-cyclopentyl-N-[2-(4-methoxypiperidin-1-yl)pyrimidin-4-yl]-1H-pyrrolo[3,2-c]pyridin-6-amine, ACETATE ION, Cyclin-dependent kinase 2 Authors: Eigenbrot, C, Yin, J. Deposit date: 2014-10-08 Release date: 2014-11-26 Last modified: 2024-11-06 Method: X-RAY DIFFRACTION (1.63 Å) Cite: Discovery of Selective and Noncovalent Diaminopyrimidine-Based Inhibitors of Epidermal Growth Factor Receptor Containing the T790M Resistance Mutation. J.Med.Chem., 57, 2014
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2014-10-08
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