Copper-Catalyzed Regio- and Stereoselective Aminoboration of Alkenylboronates
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https://figshare.com/articles/dataset/Copper-Catalyzed_Regio-_and_Stereoselective_Aminoboration_of_Alkenylboronates/3840378
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资源简介：
A copper-catalyzed
aminoboration of alkenyl dan boronates (dan
= 1,8-diaminonaphthyl) with diboron reagents and hydroxylamines
has been developed. The reaction proceeds regio- and stereoselectively
to form the corresponding β-boryl-α-aminoboronic acid
derivatives of potent interest in medicinal chemistry. Additionally,
the ligand-controlled syn/anti diastereoselectivity
switching and preliminary asymmetric catalysis are also described.
创建时间：
2016-10-03
