five

Structure of human G9a SET-domain (EHMT2) in complex with inhibitor 13

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Protein Data Bank Japan2023-10-04 更新2026-03-21 收录
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Structure of human G9a SET-domain (EHMT2) in complex with inhibitor 13 Descriptor: 6,7-dimethoxy-N~2~-methyl-N~4~-(1-methylpiperidin-4-yl)-N~2~-propylquinazoline-2,4-diamine, Histone-lysine N-methyltransferase EHMT2, S-ADENOSYLMETHIONINE, ... Authors: Babault, N, Xiong, Y, Liu, J, Jin, J. Deposit date: 2017-05-11 Release date: 2017-07-12 Last modified: 2023-10-04 Method: X-RAY DIFFRACTION (1.4 Å) Cite: Structure-activity relationship studies of G9a-like protein (GLP) inhibitors. Bioorg. Med. Chem., 25, 2017
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2017-05-11
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