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Homo sapiens Prolyl-tRNA Synthetase (HsPRS) in Complex with L-proline and compound L96

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Protein Data Bank Japan2023-11-29 更新2026-03-21 收录
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Homo sapiens Prolyl-tRNA Synthetase (HsPRS) in Complex with L-proline and compound L96 Descriptor: 4-[(3S)-3-cyano-3-cyclopropyl-2-oxidanylidene-pyrrolidin-1-yl]-N-[[3-fluoranyl-5-(5-methoxypyridin-3-yl)phenyl]methyl]-6-methyl-pyridine-2-carboxamide, Bifunctional glutamate/proline--tRNA ligase, CALCIUM ION, ... Authors: Malhotra, N, Manickam, Y, Sharma, A. Deposit date: 2021-07-04 Release date: 2022-07-06 Last modified: 2023-11-29 Method: X-RAY DIFFRACTION (2.196 Å) Cite: Targeting prolyl-tRNA synthetase via a series of ATP-mimetics to accelerate drug discovery against toxoplasmosis. Plos Pathog., 19, 2023
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2021-07-04
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