N-terminal bromodomain of human BRD2 in complex with 4,4'-(quinoline-5,7-diyl)bis(3,5-dimethylisoxazole) inhibitor
收藏Protein Data Bank Japan2024-03-13 更新2026-03-21 收录
下载链接：
https://pdbj.org/mine/summary/6mo8
下载链接
链接失效反馈官方服务：
资源简介：
N-terminal bromodomain of human BRD2 in complex with 4,4'-(quinoline-5,7-diyl)bis(3,5-dimethylisoxazole) inhibitor Descriptor: 5,7-bis(3,5-dimethyl-1,2-oxazol-4-yl)quinoline, Bromodomain-containing protein 2, SULFATE ION Authors: Lansdon, E.B, Newby, Z.E.R. Deposit date: 2018-10-04 Release date: 2019-01-23 Last modified: 2024-03-13 Method: X-RAY DIFFRACTION (1.8 Å) Cite: Structure-guided discovery of a novel, potent, and orally bioavailable 3,5-dimethylisoxazole aryl-benzimidazole BET bromodomain inhibitor. Bioorg. Med. Chem., 27, 2019
创建时间：
2018-10-04
