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Crystal structure of BRD9 bromodomain in complex with compound EA-89

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Protein Data Bank Japan2024-01-31 更新2026-03-28 收录
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Crystal structure of BRD9 bromodomain in complex with compound EA-89 Descriptor: Bromodomain-containing protein 9, ~{N}-[1,1-bis(oxidanylidene)thian-4-yl]-7-[3-methyl-1-(piperidin-4-ylmethyl)indol-5-yl]-4-oxidanylidene-5-propyl-thieno[3,2-c]pyridine-2-carboxamide Authors: Faller, M, Zink, F. Deposit date: 2022-06-21 Release date: 2022-08-10 Last modified: 2024-01-31 Method: X-RAY DIFFRACTION (1.76 Å) Cite: BRD9 degraders as chemosensitizers in acute leukemia and multiple myeloma. Blood Cancer J, 12, 2022
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2022-06-21
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