PPARgamma ligand-binding domain in complex with PG08-NL and rosiglitazone
收藏Protein Data Bank Japan2025-12-03 更新2026-04-19 收录
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https://pdbj.org/mine/summary/9v8h
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PPARgamma ligand-binding domain in complex with PG08-NL and rosiglitazone Descriptor: 2,4-THIAZOLIDIINEDIONE, 5-[[4-[2-(METHYL-2-PYRIDINYLAMINO)ETHOXY]PHENYL]METHYL]-(9CL), DI(HYDROXYETHYL)ETHER, ... Authors: Sigal, M, Okada, C, Katoh, T, Suga, H, Sengoku, T. Deposit date: 2025-05-29 Release date: 2025-11-05 Last modified: 2025-12-03 Method: X-RAY DIFFRACTION (1.39 Å) Cite: De Novo Discovery of alpha , alpha-Disubstituted alpha-amino Acid-Containing alpha-helical Peptides as Competitive PPAR gamma PPI Inhibitors. J.Am.Chem.Soc., 147, 2025
创建时间:
2025-05-29



