Crystal structure of DYRK2 in complex with EHT 5372 (Compound 1)
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Crystal structure of DYRK2 in complex with EHT 5372 (Compound 1) Descriptor: 1,2-ETHANEDIOL, Dual specificity tyrosine-phosphorylation-regulated kinase 2, methyl 9-[(2,4-dichlorophenyl)amino]-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidate Authors: Chaikuad, A, von Delft, F, Arrowsmith, C.H, Edwards, A, Bountra, C, Besson, T, Knapp, S, Structural Genomics Consortium (SGC) Deposit date: 2016-09-20 Release date: 2016-10-26 Last modified: 2024-11-20 Method: X-RAY DIFFRACTION (2.15 Å) Cite: An Unusual Binding Model of the Methyl 9-Anilinothiazolo[5,4-f] quinazoline-2-carbimidates (EHT 1610 and EHT 5372) Confers High Selectivity for Dual-Specificity Tyrosine Phosphorylation-Regulated Kinases. J. Med. Chem., 59, 2016
创建时间：
2016-09-20
