Structure of CHK1 10-pt. mutant complex with LRRK2 indazole inhibitor compound 6
收藏Protein Data Bank Japan2024-10-02 更新2026-06-30 收录
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Structure of CHK1 10-pt. mutant complex with LRRK2 indazole inhibitor compound 6 Descriptor: (1S,4r)-4-[(1P)-5-chloro-1-(1-methyl-1H-pyrazol-4-yl)-1H-indazol-6-yl]-1-(oxetan-3-yl)piperidin-1-ium, 1,2-ETHANEDIOL, Serine/threonine-protein kinase Chk1 Authors: Palte, R.L, Zebisch, M, Henry, C, Barker, J.J. Deposit date: 2024-06-26 Release date: 2024-09-18 Last modified: 2024-10-02 Method: X-RAY DIFFRACTION (1.31 Å) Cite: Discovery and Optimization of N-Heteroaryl Indazole LRRK2 Inhibitors. J.Med.Chem., 67, 2024
创建时间:
2024-06-26



