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Crystal structure of the first bromodomain of human BRD4 in complex with MS417 inhibitor

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Protein Data Bank Japan2023-09-13 更新2026-03-21 收录
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Crystal structure of the first bromodomain of human BRD4 in complex with MS417 inhibitor Descriptor: 1,2-ETHANEDIOL, Bromodomain-containing protein 4, methyl [(6S)-4-(4-chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepin-6-yl]acetate Authors: Joshua, J, Zhou, M.-M, Plotnikov, A.N. Deposit date: 2012-05-09 Release date: 2012-09-12 Last modified: 2023-09-13 Method: X-RAY DIFFRACTION (1.4 Å) Cite: Down-regulation of NF-{kappa}B Transcriptional Activity in HIV-associated Kidney Disease by BRD4 Inhibition. J.Biol.Chem., 287, 2012
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2012-05-09
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