Crystal structure of HIV-1 protease in complex with macrocyclic peptide
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Crystal structure of HIV-1 protease in complex with macrocyclic peptide Descriptor: MAGNESIUM ION, Macrocyclic Peptide, Protease Authors: Kusumoto, Y, Sato, S, Yamada, T, Kozono, I, Nakata, Z, Asada, N, Mitsuki, S, Wakasa-Morimoto, C, Tohru, M, Watanabe, A, Hayashi, K, Mikamiyama, H. Deposit date: 2022-07-07 Release date: 2022-11-02 Last modified: 2024-11-13 Method: X-RAY DIFFRACTION (2.01 Å) Cite: Highly Potent and Oral Macrocyclic Peptides as a HIV-1 Protease Inhibitor: mRNA Display-Derived Hit-to-Lead Optimization. Acs Med.Chem.Lett., 13, 2022
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2022-07-07



