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Crystal structure of human DHODH in complex with BAY 2402234

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Protein Data Bank Japan2024-05-15 更新2026-03-21 收录
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Crystal structure of human DHODH in complex with BAY 2402234 Descriptor: ACETATE ION, Dihydroorotate dehydrogenase (quinone), mitochondrial, ... Authors: Friberg, A, Gradl, S. Deposit date: 2019-02-26 Release date: 2019-06-05 Last modified: 2024-05-15 Method: X-RAY DIFFRACTION (1.52 Å) Cite: The novel dihydroorotate dehydrogenase (DHODH) inhibitor BAY 2402234 triggers differentiation and is effective in the treatment of myeloid malignancies. Leukemia, 33, 2019
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2019-02-26
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