five

SARS-CoV-2 papain-like protease (PLpro) with inhibitor Jun12199

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Protein Data Bank Japan2024-05-01 更新2026-04-19 收录
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https://pdbj.org/mine/summary/8uuh
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SARS-CoV-2 papain-like protease (PLpro) with inhibitor Jun12199 Descriptor: 5-[2-(dimethylamino)ethoxy]-2-methyl-N-[(1R)-1-{(3M,5P)-3-(1-methyl-1H-pyrazol-4-yl)-5-[1-(propan-2-yl)-1H-pyrazol-4-yl]phenyl}ethyl]benzamide, CHLORIDE ION, DI(HYDROXYETHYL)ETHER, ... Authors: Ansari, A, Tan, B, Ruiz, F.X, Arnold, E, Wang, J. Deposit date: 2023-11-01 Release date: 2024-04-03 Last modified: 2024-05-01 Method: X-RAY DIFFRACTION (2.8 Å) Cite: Design of a SARS-CoV-2 papain-like protease inhibitor with antiviral efficacy in a mouse model. Science, 383, 2024
创建时间:
2023-11-01
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