Crystal structure of the first bromodomain (BD1) of human BRDT bound to LRRK2-IN-1
收藏Protein Data Bank Japan2023-10-18 更新2026-03-21 收录
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Crystal structure of the first bromodomain (BD1) of human BRDT bound to LRRK2-IN-1 Descriptor: 1,2-ETHANEDIOL, 2-[(2-methoxy-4-{[4-(4-methylpiperazin-1-yl)piperidin-1-yl]carbonyl}phenyl)amino]-5,11-dimethyl-5,11-dihydro-6H-pyrimido[4,5-b][1,4]benzodiazepin-6-one, Bromodomain testis-specific protein Authors: Chan, A, Karim, M.R, Schonbrunn, E. Deposit date: 2021-01-14 Release date: 2021-07-14 Last modified: 2023-10-18 Method: X-RAY DIFFRACTION (1.89 Å) Cite: Differential BET Bromodomain Inhibition by Dihydropteridinone and Pyrimidodiazepinone Kinase Inhibitors. J.Med.Chem., 64, 2021
创建时间:
2021-01-14



