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Structure of human ATAD2 bromodomain bound to fragment inhibitor

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Protein Data Bank Japan2023-09-27 更新2026-03-21 收录
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Structure of human ATAD2 bromodomain bound to fragment inhibitor Descriptor: 2-amino-7,7-dimethyl-5,6,7,8-tetrahydro-4H-[1,3]thiazolo[5,4-c]azepin-4-one, ATPase family AAA domain-containing protein 2, CHLORIDE ION, ... Authors: Harner, M.J, Chauder, B.A, Phan, J, Fesik, S.W. Deposit date: 2014-07-09 Release date: 2014-10-29 Last modified: 2023-09-27 Method: X-RAY DIFFRACTION (2.15 Å) Cite: Fragment-Based Screening of the Bromodomain of ATAD2. J.Med.Chem., 57, 2014

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2014-07-09
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