novel orally efficacious inhibitors complexed with PARP1
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novel orally efficacious inhibitors complexed with PARP1 Descriptor: 6-fluoranyl-2-(4,5,6,7-tetrahydrothieno[3,2-c]pyridin-2-yl)-1~{H}-benzimidazole-4-carboxamide, Poly [ADP-ribose] polymerase 1, SULFATE ION Authors: Liu, Q, Xu, Y. Deposit date: 2017-06-15 Release date: 2018-04-25 Last modified: 2024-10-16 Method: X-RAY DIFFRACTION (2.3 Å) Cite: Design and synthesis of 2-(4,5,6,7-tetrahydrothienopyridin-2-yl)-benzoimidazole carboxamides as novel orally efficacious Poly(ADP-ribose)polymerase (PARP) inhibitors Eur J Med Chem, 145, 2018
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2017-06-15



