five

EGFR kinase domain mutant "TMLR" with a pyrazolopyrimidine inhibitor

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Protein Data Bank Japan2024-03-06 更新2026-03-21 收录
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https://pdbj.org/mine/summary/5hib
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资源简介:
EGFR kinase domain mutant "TMLR" with a pyrazolopyrimidine inhibitor Descriptor: Epidermal growth factor receptor, N-tert-butyl-5-{[(1-methyl-1H-pyrazol-5-yl)sulfonyl]amino}pyrazolo[1,5-a]pyrimidine-3-carboxamide Authors: Eigenbrot, C, Yu, C. Deposit date: 2016-01-11 Release date: 2016-04-06 Last modified: 2024-03-06 Method: X-RAY DIFFRACTION (2.85 Å) Cite: Activation Mechanism of Oncogenic Deletion Mutations in BRAF, EGFR, and HER2. Cancer Cell, 29, 2016
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2016-01-11
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