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Leishmania major N-myristoyltransferase in complex with thienopyrimidine inhibitor IMP-0000105

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Protein Data Bank Japan2024-05-15 更新2026-03-21 收录
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https://pdbj.org/mine/summary/6qdd
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Leishmania major N-myristoyltransferase in complex with thienopyrimidine inhibitor IMP-0000105 Descriptor: 2-[(2~{S})-1-[2-[methyl-(1-methylpiperidin-4-yl)amino]thieno[3,2-d]pyrimidin-4-yl]-2,3-dihydropyrrol-2-yl]ethanenitrile, DIMETHYL SULFOXIDE, Glycylpeptide N-tetradecanoyltransferase, ... Authors: Brannigan, J.A. Deposit date: 2019-01-01 Release date: 2020-05-06 Last modified: 2024-05-15 Method: X-RAY DIFFRACTION (1.65 Å) Cite: Novel Thienopyrimidine Inhibitors of Leishmania N -Myristoyltransferase with On-Target Activity in Intracellular Amastigotes. J.Med.Chem., 63, 2020
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2019-01-01
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