Aurora A kinase domain with phthalazinone pyrazole inhibitor
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Aurora A kinase domain with phthalazinone pyrazole inhibitor Descriptor: 4-[(5-methyl-1H-pyrazol-3-yl)amino]-2-phenylphthalazin-1(2H)-one, Serine/threonine-protein kinase 6 Authors: Kairies, N.A, Oliveira, T, Engh, R.A. Deposit date: 2010-10-17 Release date: 2011-03-23 Last modified: 2024-02-21 Method: X-RAY DIFFRACTION (2.8 Å) Cite: Phthalazinone pyrazoles as potent, selective, and orally bioavailable inhibitors of aurora-a kinase. J.Med.Chem., 54, 2011
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2010-10-17



