PORCINE PANCREATIC ELASTASE COMPLEXED WITH GW311616A
收藏Protein Data Bank Japan2024-11-13 更新2026-03-21 收录
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https://pdbj.org/mine/summary/1hv7
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PORCINE PANCREATIC ELASTASE COMPLEXED WITH GW311616A Descriptor: ELASTASE 1, N-[2-(1-FORMYL-2-METHYL-PROPYL)-1-(4-PIPERIDIN-1-YL-BUT-2-ENOYL)-PYRROLIDIN-3-YL]-METHANESULFONAMIDE, SULFATE ION Authors: Skarzynski, T, Singh, O.M. Deposit date: 2001-01-08 Release date: 2001-01-17 Last modified: 2024-11-13 Method: X-RAY DIFFRACTION (1.7 Å) Cite: The discovery of a potent, intracellular, orally bioavailable, long duration inhibitor of human neutrophil elastase--GW311616A a development candidate Bioorg.Med.Chem.Lett., 11, 2001
创建时间:
2001-01-08



