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Human steroidogenic cytochrome P450 17A1 mutant N52Y with inhibitor abiraterone

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Protein Data Bank Japan2024-04-03 更新2026-03-21 收录
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https://pdbj.org/mine/summary/6wr1
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Human steroidogenic cytochrome P450 17A1 mutant N52Y with inhibitor abiraterone Descriptor: Abiraterone, PROTOPORPHYRIN IX CONTAINING FE, Steroid 17-alpha-hydroxylase/17,20 lyase Authors: Petrunak, E.M, Bart, A.G, Scott, E.E. Deposit date: 2020-04-29 Release date: 2021-05-05 Last modified: 2024-04-03 Method: X-RAY DIFFRACTION (1.85 Å) Cite: Human cytochrome P450 17A1 structures with metabolites of prostate cancer drug abiraterone reveal substrate-binding plasticity and a second binding site. J.Biol.Chem., 299, 2023
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2020-04-29
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