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Crystal structure of the human BRPF1 bromodomain in complex with BZ038

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Protein Data Bank Japan2024-01-17 更新2026-03-21 收录
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Crystal structure of the human BRPF1 bromodomain in complex with BZ038 Descriptor: 1-ethyl-~{N}-[(~{R})-(3-fluorophenyl)-(1-methylimidazol-2-yl)methyl]-2,3-bis(oxidanylidene)-4~{H}-quinoxaline-6-carboxamide, NITRATE ION, Peregrin Authors: Zhu, J, Caflisch, A. Deposit date: 2017-06-01 Release date: 2018-06-13 Last modified: 2024-01-17 Method: X-RAY DIFFRACTION (1.302 Å) Cite: Structure-based discovery of selective BRPF1 bromodomain inhibitors. Eur J Med Chem, 155, 2018
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2017-06-01
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