遇见数据集

JAK2 Pseudokinase in complex with BI-D1870

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Protein Data Bank Japan2024-03-13 更新2026-03-21 收录
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JAK2 Pseudokinase in complex with BI-D1870 Descriptor: (7R)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(3-methylbutyl)-7,8-dihydropteridin-6(5H)-one, Tyrosine-protein kinase JAK2 Authors: Li, Q, Eck, M.J, Li, K, Park, E. Deposit date: 2017-07-19 Release date: 2018-08-01 Last modified: 2024-03-13 Method: X-RAY DIFFRACTION (2.6 Å) Cite: Discovery and Structural Characterization of ATP-Site Ligands for the Wild-Type and V617F Mutant JAK2 Pseudokinase Domain. ACS Chem. Biol., 14, 2019

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2017-07-19
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