M3 muscarinic acetylcholine receptor in complex with a selective antagonist
收藏Protein Data Bank Japan2024-11-20 更新2026-03-21 收录
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M3 muscarinic acetylcholine receptor in complex with a selective antagonist Descriptor: (1R,2R,4S,5S,7s)-7-({[4-fluoro-2-(thiophen-2-yl)phenyl]carbamoyl}oxy)-9,9-dimethyl-3-oxa-9-azatricyclo[3.3.1.0~2,4~]nonan-9-ium, CITRIC ACID, HEXAETHYLENE GLYCOL, ... Authors: Liu, H, Hofmann, J, Fish, I, Schaake, B, Eitel, K, Bartuschat, A, Kaindl, J, Rampp, H, Banerjee, A, Hubner, H, Clark, M.J, Vincent, S.G, Fisher, J, Heinrich, M, Hirata, K, Liu, X, Sunahara, R.K, Shoichet, B.K, Kobilka, B.K, Gmeiner, P. Deposit date: 2018-03-13 Release date: 2018-11-28 Last modified: 2024-11-20 Method: X-RAY DIFFRACTION (3.1 Å) Cite: Structure-guided development of selective M3 muscarinic acetylcholine receptor antagonists Proc. Natl. Acad. Sci. U.S.A., 115, 2018
创建时间:
2018-03-13



