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Crystal Structure of human PARP-1 CAT domain bound to inhibitor UKTT15

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Protein Data Bank Japan2024-11-13 更新2026-03-21 收录
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Crystal Structure of human PARP-1 CAT domain bound to inhibitor UKTT15 Descriptor: Poly [ADP-ribose] polymerase 1, SULFATE ION, methyl 2-{4-[4-(7-carbamoyl-1H-benzimidazol-2-yl)benzene-1-carbonyl]piperazin-1-yl}pyrimidine-5-carboxylate Authors: Langelier, M.F, Pascal, J.M. Deposit date: 2020-01-21 Release date: 2020-06-17 Last modified: 2024-11-13 Method: X-RAY DIFFRACTION (2.8 Å) Cite: Structural basis for allosteric PARP-1 retention on DNA breaks. Science, 368, 2020

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2020-01-21
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