Crystal strcuture of Keap1_compound_1
收藏Protein Data Bank Japan2025-09-17 更新2026-04-19 收录
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Crystal strcuture of Keap1_compound_1 Descriptor: Kelch-like ECH-associated protein 1, ~{N},~{N}'-bis[4-[(2-azanyl-2-oxidanylidene-ethyl)-[4-[(2-azanyl-2-oxidanylidene-ethyl)-(4-methoxyphenyl)sulfonyl-amino]naphthalen-1-yl]sulfamoyl]phenyl]pentanediamide Authors: Xu, K. Deposit date: 2024-08-18 Release date: 2025-06-25 Last modified: 2025-09-17 Method: X-RAY DIFFRACTION (2.993 Å) Cite: Chemical knockdown of Keap1 and homoPROTAC-ing allergic rhinitis. Acta Pharm Sin B, 15, 2025
创建时间:
2024-08-18



