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Inhibited structure of IMPDH from Pseudomonas aeruginosa

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Protein Data Bank Japan2024-01-17 更新2026-03-21 收录
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Inhibited structure of IMPDH from Pseudomonas aeruginosa Descriptor: (5~{S})-7-azanyl-5-(4-chlorophenyl)-2,4-bis(oxidanylidene)-1,5-dihydropyrano[2,3-d]pyrimidine-6-carbonitrile, Inosine-5'-monophosphate dehydrogenase, SULFATE ION Authors: Labesse, G, Alexandre, T, Haouz, A, Munier-Lehmann, H. Deposit date: 2018-05-18 Release date: 2019-02-27 Last modified: 2024-01-17 Method: X-RAY DIFFRACTION (2.54 Å) Cite: First-in-class allosteric inhibitors of bacterial IMPDHs. Eur J Med Chem, 167, 2019

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2018-05-18
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