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Crystal structure of human Naa50 in complex with a truncated cofactor derived inhibitor (compound 2)

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Protein Data Bank Japan2024-10-23 更新2026-03-21 收录
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Crystal structure of human Naa50 in complex with a truncated cofactor derived inhibitor (compound 2) Descriptor: (2R)-2-hydroxy-3,3-dimethyl-N-{3-oxo-3-[(2-sulfanylethyl)amino]propyl}butanamide, ACE-MET-LEU-GLY-PRO-NH2, N-alpha-acetyltransferase 50 Authors: Greasley, S.E, Feng, J, Deng, Y.-L, Stewart, A.E. Deposit date: 2020-04-03 Release date: 2020-07-01 Last modified: 2024-10-23 Method: X-RAY DIFFRACTION (2.04 Å) Cite: Characterization of SpecificN-alpha-Acetyltransferase 50 (Naa50) Inhibitors Identified Using a DNA Encoded Library. Acs Med.Chem.Lett., 11, 2020
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2020-04-03
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