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Discovery of Selective BRD4 BD1 Inhibitor Based on [1,2,4] triazolo [4,3-b] pyridazine Scaffold

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Protein Data Bank Japan2023-11-29 更新2026-05-23 收录
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Discovery of Selective BRD4 BD1 Inhibitor Based on [1,2,4] triazolo [4,3-b] pyridazine Scaffold Descriptor: (2~{R})-2-[[3-methyl-6-(2-phenoxyphenyl)-[1,2,4]triazolo[4,3-b]pyridazin-8-yl]amino]propanamide, Isoform C of Bromodomain-containing protein 4 Authors: Cao, D, Xiong, B. Deposit date: 2022-03-08 Release date: 2023-03-22 Last modified: 2023-11-29 Method: X-RAY DIFFRACTION (1.44 Å) Cite: Discovery of Selective BRD4 BD1 Inhibitor Based on [1,2,4] triazolo [4,3-b] pyridazine Scaffold To Be Published

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2022-03-08
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