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Crystal structure of murine NF-kappaB inducing kinase (NIK) in complex with compound 2f

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Protein Data Bank Japan2024-01-17 更新2026-03-21 收录
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Crystal structure of murine NF-kappaB inducing kinase (NIK) in complex with compound 2f Descriptor: 5-fluoranyl-1-[4-[2-[(3~{R})-1-methyl-3-oxidanyl-2-oxidanylidene-pyrrol-3-yl]ethynyl]pyridin-2-yl]indazole-3-carboxamide, Mitogen-activated protein kinase kinase kinase 14 Authors: Leonardo-Silvestre, H, McEwan, P.A, Hymowitz, S.G. Deposit date: 2018-03-28 Release date: 2018-07-04 Last modified: 2024-01-17 Method: X-RAY DIFFRACTION (2.84 Å) Cite: Scaffold-Hopping Approach To Discover Potent, Selective, and Efficacious Inhibitors of NF-kappa B Inducing Kinase. J. Med. Chem., 61, 2018

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2018-03-28
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