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Crystal structure of the midazolam-bound human CYP3A4

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Protein Data Bank Japan2023-10-04 更新2026-03-21 收录
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Crystal structure of the midazolam-bound human CYP3A4 Descriptor: 8-chloro-6-(2-fluorophenyl)-1-methyl-4H-imidazo[1,5-a][1,4]benzodiazepine, Cytochrome P450 3A4, PROTOPORPHYRIN IX CONTAINING FE Authors: Sevrioukova, I, Poulos, T. Deposit date: 2016-09-20 Release date: 2016-12-07 Last modified: 2023-10-04 Method: X-RAY DIFFRACTION (2.7 Å) Cite: Structural basis for regiospecific midazolam oxidation by human cytochrome P450 3A4. Proc. Natl. Acad. Sci. U.S.A., 114, 2017

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2016-09-20
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