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TAS-120 covalent complex with FGFR1

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Protein Data Bank Japan2024-11-20 更新2026-03-21 收录
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资源简介:
TAS-120 covalent complex with FGFR1 Descriptor: 1-[(3S)-3-{4-amino-3-[(3,5-dimethoxyphenyl)ethynyl]-1H-pyrazolo[3,4-d]pyrimidin-1-yl}pyrrolidin-1-yl]prop-2-en-1-one, Fibroblast growth factor receptor 1, SULFATE ION Authors: Kalyukina, M, Squire, C.J. Deposit date: 2018-11-05 Release date: 2019-01-16 Last modified: 2024-11-20 Method: X-RAY DIFFRACTION (2.2 Å) Cite: TAS-120 Cancer Target Binding: Defining Reactivity and Revealing the First Fibroblast Growth Factor Receptor 1 (FGFR1) Irreversible Structure. ChemMedChem, 14, 2019
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2018-11-05
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