Crystal structure of an extender (SPD28345)-modified human PDK1 complex 2
收藏Protein Data Bank Japan2024-10-09 更新2026-03-21 收录
下载链接:
https://pdbj.org/mine/summary/3pwy
下载链接
链接失效反馈官方服务:
资源简介:
Crystal structure of an extender (SPD28345)-modified human PDK1 complex 2 Descriptor: 3-phosphoinositide-dependent protein kinase 1, N-[2-({6-[(2-sulfanylethyl)amino]pyrimidin-4-yl}amino)ethyl]propanamide Authors: Elling, R.A, Penny, D.M, Simmons, R.L, Erlanson, D.A, Romanowski, M.J. Deposit date: 2010-12-09 Release date: 2011-04-20 Last modified: 2024-10-09 Method: X-RAY DIFFRACTION (3.5 Å) Cite: Discovery of a potent and highly selective PDK1 inhibitor via fragment-based drug discovery. Bioorg.Med.Chem.Lett., 21, 2011
创建时间:
2010-12-09



