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Toxoplasma Gondii CDPK1 in complex with inhibitor GXJ-186

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Protein Data Bank Japan2026-05-20 更新2026-03-21 收录
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https://pdbj.org/mine/summary/5w9e
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Toxoplasma Gondii CDPK1 in complex with inhibitor GXJ-186 Descriptor: 1-tert-butyl-3-[(3-chlorophenyl)sulfanyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine, Calmodulin-domain protein kinase 1 Authors: El Bakkouri, M, Lovato, D, Loppnau, P, Lin, Y.H, Rutaganaria, F, Lopez, M.S, Shokat, L, Bountra, C, Edwards, A.M, Arrowsmith, C.H, Sibley, D, Hui, R, Walker, J.R. Deposit date: 2017-06-23 Release date: 2017-08-02 Last modified: 2026-05-20 Method: X-RAY DIFFRACTION (2.44 Å) Cite: Inhibition of Calcium Dependent Protein Kinase 1 (CDPK1) by Pyrazolopyrimidine Analogs Decreases Establishment and Reoccurrence of Central Nervous System Disease by Toxoplasma gondii. J.Med.Chem., 60, 2017
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2017-06-23
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