five

RORgamma in complex with agonist BIO592 and Coactivator EBI96

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Protein Data Bank Japan2024-10-23 更新2026-03-21 收录
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RORgamma in complex with agonist BIO592 and Coactivator EBI96 Descriptor: CHLORIDE ION, GLU-PHE-PRO-TYR-LEU-LEU-SER-LEU-LEU-GLY-GLU-VAL-SER-PRO-GLN, N-(4-ethyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)-3,4-dimethyl-N-(2,2,2-trifluoroethyl)benzene-1-sulfonamide, ... Authors: Marcotte, D.J. Deposit date: 2016-03-24 Release date: 2016-06-15 Last modified: 2024-10-23 Method: X-RAY DIFFRACTION (2.635 Å) Cite: Structural determinant for inducing RORgamma specific inverse agonism triggered by a synthetic benzoxazinone ligand. Bmc Struct.Biol., 16, 2016
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2016-03-24
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