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BRD4 Bromodomain 1 in complex with multi-action inhibitor SRX3212

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Protein Data Bank Japan2023-10-18 更新2026-03-21 收录
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https://pdbj.org/mine/summary/6x7c
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BRD4 Bromodomain 1 in complex with multi-action inhibitor SRX3212 Descriptor: 7-[5-(morpholin-4-yl)-7-oxo-7H-thieno[3,2-b]pyran-3-yl]-N-[(pyridin-3-yl)methyl]-2,3-dihydro-1,4-benzodioxine-5-carboxamide, Bromodomain-containing protein 4 Authors: Vann, K.R, Kutateladze, T.G. Deposit date: 2020-05-29 Release date: 2020-08-05 Last modified: 2023-10-18 Method: X-RAY DIFFRACTION (2.7 Å) Cite: Design of thienopyranone-based BET inhibitors that bind multiple synthetic lethality targets. Sci Rep, 10, 2020
创建时间:
2020-05-29
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