five

Human FGFR1 kinase in complex with CH5183284

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Protein Data Bank Japan2023-11-08 更新2026-03-21 收录
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资源简介:
Human FGFR1 kinase in complex with CH5183284 Descriptor: Fibroblast growth factor receptor 1, SULFATE ION, [5-amino-1-(2-methyl-1H-benzimidazol-6-yl)-1H-pyrazol-4-yl](1H-indol-2-yl)methanone Authors: Fukami, T.A, Lukacs, C.M, Janson, C. Deposit date: 2016-06-09 Release date: 2016-06-22 Last modified: 2023-11-08 Method: X-RAY DIFFRACTION (2.15 Å) Cite: The fibroblast growth factor receptor genetic status as a potential predictor of the sensitivity to CH5183284/Debio 1347, a novel selective FGFR inhibitor Mol.Cancer Ther., 13, 2014
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2016-06-09
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