遇见数据集

USP7 IN COMPLEX WITH LIGAND COMPOUND 23

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Protein Data Bank Japan2024-10-30 更新2026-03-21 收录
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USP7 IN COMPLEX WITH LIGAND COMPOUND 23 Descriptor: 1-{[7-(5-chloro-2-{[(3R,4S)-4-fluoropyrrolidin-3-yl]oxy}-3-methylphenyl)thieno[3,2-b]pyridin-2-yl]methyl}-1H-pyrrole-2,5-dione, Ubiquitin carboxyl-terminal hydrolase 7 Authors: Leger, P.R, Wustrow, D.J, Hu, D.X, Krapp, S, Maskos, K, Blaesse, M. Deposit date: 2020-01-29 Release date: 2020-04-29 Last modified: 2024-10-30 Method: X-RAY DIFFRACTION (2.73 Å) Cite: Discovery of Potent, Selective, and Orally Bioavailable Inhibitors of USP7 with In Vivo Antitumor Activity. J.Med.Chem., 63, 2020

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2020-01-29
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