Bovine GRK2 in complex with Gbetagamma subunits and a selective kinase inhibitor (CMPD101)
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Bovine GRK2 in complex with Gbetagamma subunits and a selective kinase inhibitor (CMPD101) Descriptor: 3-({[4-methyl-5-(pyridin-4-yl)-4H-1,2,4-triazol-3-yl]methyl}amino)-N-[2-(trifluoromethyl)benzyl]benzamide, Beta-adrenergic receptor kinase 1, Guanine nucleotide-binding protein G(I)/G(S)/G(O) subunit gamma-2, ... Authors: Thal, D.M, Tesmer, J.J. Deposit date: 2010-12-07 Release date: 2011-06-01 Last modified: 2023-09-06 Method: X-RAY DIFFRACTION (2.48 Å) Cite: Molecular Mechanism of Selectivity among G Protein-Coupled Receptor Kinase 2 Inhibitors. Mol.Pharmacol., 80, 2011
创建时间:
2010-12-07



