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BACE crystal structure with tricyclic aminothiazine inhibitor

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Protein Data Bank Japan2024-10-30 更新2026-03-21 收录
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BACE crystal structure with tricyclic aminothiazine inhibitor Descriptor: Beta-secretase 1, N-[(4aS,6S,8aR)-2-amino-5,6,7,8-tetrahydro-4a,8a-(methanooxymethano)-3,1-benzothiazin-6(4H)-yl]-3-chlorobenzamide Authors: Timm, D.E. Deposit date: 2015-05-13 Release date: 2015-06-10 Last modified: 2024-10-30 Method: X-RAY DIFFRACTION (1.65 Å) Cite: Preparation and biological evaluation of conformationally constrained BACE1 inhibitors. Bioorg.Med.Chem., 23, 2015

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2015-05-13
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