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Tankyrase 2 catalytic domain in complex with OUL40

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Protein Data Bank Japan2024-02-07 更新2026-04-19 收录
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Tankyrase 2 catalytic domain in complex with OUL40 Descriptor: 6-methyl-[1,2,4]triazolo[3,4-b][1,3]benzothiazole, GLYCEROL, Poly [ADP-ribose] polymerase tankyrase-2, ... Authors: Murthy, S, Venkannagari, H, Maksimainen, M.M, Lehtio, L. Deposit date: 2022-02-08 Release date: 2023-01-25 Last modified: 2024-02-07 Method: X-RAY DIFFRACTION (2.25 Å) Cite: [1,2,4]Triazolo[3,4- b ]benzothiazole Scaffold as Versatile Nicotinamide Mimic Allowing Nanomolar Inhibition of Different PARP Enzymes. J.Med.Chem., 66, 2023

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2022-02-08
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