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HIV-1 PROTEASE IN COMPLEX WITH A DIFLUOROKETONE CONTAINING INHIBITOR A79285

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Protein Data Bank Japan2024-06-05 更新2026-03-21 收录
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https://pdbj.org/mine/summary/1dif
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HIV-1 PROTEASE IN COMPLEX WITH A DIFLUOROKETONE CONTAINING INHIBITOR A79285 Descriptor: BETA-MERCAPTOETHANOL, HIV-1 PROTEASE, N-{1-BENZYL-2,2-DIFLUORO-3,3-DIHYDROXY-4-[3-METHYL-2-(3-METHYL-3-PYRIDIN-2-YLMETHYL-UREIDO)-BUTYRYLAMINO]-5-PHENYL-PENTYL}-3-METHYL-2-(3-METHYL-3-PYRIDIN-2-YLMETHYL-UREIDO)-BUTYRAMIDE Authors: Silva, A.M, Cachau, R.E, Sham, H.L, Erickson, J.W. Deposit date: 1995-10-09 Release date: 1996-03-08 Last modified: 2024-06-05 Method: X-RAY DIFFRACTION (1.7 Å) Cite: Inhibition and catalytic mechanism of HIV-1 aspartic protease. J.Mol.Biol., 255, 1996
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1995-10-09
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