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Crystal structure of NS3/4A protease variant R155K in complex with danoprevir

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Protein Data Bank Japan2023-09-13 更新2026-03-21 收录
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Crystal structure of NS3/4A protease variant R155K in complex with danoprevir Descriptor: (2R,6S,12Z,13aS,14aR,16aS)-6-[(tert-butoxycarbonyl)amino]-14a-[(cyclopropylsulfonyl)carbamoyl]-5,16-dioxo-1,2,3,5,6,7,8 ,9,10,11,13a,14,14a,15,16,16a-hexadecahydrocyclopropa[e]pyrrolo[1,2-a][1,4]diazacyclopentadecin-2-yl 4-fluoro-2H-isoindole-2-carboxylate, Genome polyprotein, SULFATE ION, ... Authors: Schiffer, C.A, Romano, K.P. Deposit date: 2011-07-11 Release date: 2012-09-05 Last modified: 2023-09-13 Method: X-RAY DIFFRACTION (1.159 Å) Cite: The Molecular Basis of Drug Resistance against Hepatitis C Virus NS3/4A Protease Inhibitors. Plos Pathog., 8, 2012
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2011-07-11
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