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Crystal structure of TD1-gatorbulin1 complex

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Protein Data Bank Japan2024-01-31 更新2026-03-21 收录
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Crystal structure of TD1-gatorbulin1 complex Descriptor: (2~{R})-2-oxidanyl-2-[(6~{S},9~{S},12~{S},15~{S},17~{S})-6,10,12,17-tetramethyl-3-methylidene-7-oxidanyl-2,5,8,11,14-pentakis(oxidanylidene)-13-oxa-1,4,7,10-tetrazabicyclo[13.3.0]octadecan-9-yl]ethanamide, Designed Ankyrin Repeat Protein (DARPIN) D1, GLYCEROL, ... Authors: Oliva, M.A, Diaz, J.F. Deposit date: 2020-10-07 Release date: 2021-03-03 Last modified: 2024-01-31 Method: X-RAY DIFFRACTION (1.93 Å) Cite: Gatorbulin-1, a distinct cyclodepsipeptide chemotype, targets a seventh tubulin pharmacological site. Proc.Natl.Acad.Sci.USA, 118, 2021
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2020-10-07
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