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Structure-guided discovery of selective USP7 inhibitors with in vivo activity

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Protein Data Bank Japan2024-11-27 更新2026-04-19 收录
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Structure-guided discovery of selective USP7 inhibitors with in vivo activity Descriptor: 3-[[1-[(3~{R},4~{R})-1-[5-(3-methoxypyridin-4-yl)thiophen-2-yl]carbonyl-3-phenyl-piperidin-4-yl]carbonyl-4-oxidanyl-piperidin-4-yl]methyl]-7-methyl-pyrrolo[2,3-d]pyrimidin-4-one, Ubiquitin carboxyl-terminal hydrolase 7 Authors: Baker, L.M, Murray, J, Hubbard, R.E, Whitehead, N. Deposit date: 2024-05-29 Release date: 2024-11-06 Last modified: 2024-11-27 Method: X-RAY DIFFRACTION (3.37 Å) Cite: Structure-Guided Discovery of Selective USP7 Inhibitors with In Vivo Activity. J.Med.Chem., 67, 2024
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2024-05-29
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