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Bcl-xL in complex with inhibitor (Compound 10)

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Protein Data Bank Japan2023-12-27 更新2026-03-21 收录
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Bcl-xL in complex with inhibitor (Compound 10) Descriptor: 1,2-ETHANEDIOL, 2-[8-(1,3-benzothiazol-2-ylcarbamoyl)-3,4-dihydroisoquinolin-2(1H)-yl]-5-{3-[4-(1H-pyrazolo[3,4-d]pyrimidin-1-yl)phenoxy]propyl}-1,3-thiazole-4-carboxylic acid, ACETATE ION, ... Authors: Czabotar, P.E, Lessense, G, Smith, B.J, Colman, P.M. Deposit date: 2014-06-24 Release date: 2014-10-15 Last modified: 2023-12-27 Method: X-RAY DIFFRACTION (1.8 Å) Cite: Structure-Guided Rescaffolding of Selective Antagonists of BCL-XL. Acs Med.Chem.Lett., 5, 2014

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2014-06-24
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