N-TERMINAL BROMODOMAIN OF HUMAN BRD4 with I-BET567
收藏Protein Data Bank Japan2024-05-01 更新2026-04-19 收录
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https://pdbj.org/mine/summary/7qdl
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N-TERMINAL BROMODOMAIN OF HUMAN BRD4 with I-BET567 Descriptor: (2S,4R)-1-acetyl-4-((5-chloropyrimidin-2-yl)amino)-2-methyl-1,2,3,4-tetrahydroquinoline-6-carboxamide, 1,2-ETHANEDIOL, Bromodomain-containing protein 4 Authors: Chung, C. Deposit date: 2021-11-27 Release date: 2022-12-14 Last modified: 2024-05-01 Method: X-RAY DIFFRACTION (1.67 Å) Cite: Design, Synthesis, and Characterization of I-BET567, a Pan-Bromodomain and Extra Terminal (BET) Bromodomain Oral Candidate. J.Med.Chem., 65, 2022
创建时间:
2021-11-27



